The Effect of MK0859 on Lipoprotein Metabolism in Patients With Dyslipidemia (0859-026 AM3)
Primary Purpose
Dyslipidemia
Status
Completed
Phase
Phase 1
Locations
Study Type
Interventional
Intervention
anacetrapib
Comparator: atorvastatin
Comparator: placebo to MK0859
Comparator: placebo to atorvastatin
Sponsored by
About this trial
This is an interventional treatment trial for Dyslipidemia
Eligibility Criteria
Inclusion Criteria:
- Patient's weight has been stable for at least 6 weeks
- Patient is in good health based on medical history, physical exam, and laboratory tests
- Patient has dyslipidemia
Exclusion Criteria :
- Patient has a history of stroke, seizures, or major neurological disorders
- Patient has a history of cancer
- Patient is currently taking any lipid-lowering medications or substances except for statins
- Patient consumes excessive amounts of alcohol or caffeine
- Patient has multiple and/or severe allergies to food or drugs
Sites / Locations
Arms of the Study
Arm 1
Arm 2
Arm Type
Experimental
Experimental
Arm Label
Panel A
Panel B
Arm Description
Period 1: atorvastatin + placebo to MK0859; Period 2: atorvastatin + MK0859
Period 1: placebo to atorvastatin + placebo to MK0859; Period 2: MK0859 + placebo to atorvastatin
Outcomes
Primary Outcome Measures
Difference in Production Rate (PR) and Fractional Catabolic Rate (FCR) of Low Density Lipoprotein (LDL) apoB100 following treatment with MK0859 and atorvastatin versus atorvastatin alone
Secondary Outcome Measures
Difference in FCR of LDL apoB100 following treatment with MK0859 versus placebo
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT00990808
Brief Title
The Effect of MK0859 on Lipoprotein Metabolism in Patients With Dyslipidemia (0859-026 AM3)
Official Title
A Multiple Dose Study to Investigate the Effect of MK0859 on Lipoprotein Metabolism When Added to Ongoing Statin Therapy in Dyslipidemic Patients
Study Type
Interventional
2. Study Status
Record Verification Date
June 2015
Overall Recruitment Status
Completed
Study Start Date
November 2009 (undefined)
Primary Completion Date
June 2011 (Actual)
Study Completion Date
July 2011 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Merck Sharp & Dohme LLC
4. Oversight
Data Monitoring Committee
No
5. Study Description
Brief Summary
This study will investigate the effect of MK0859 on lipoprotein metabolism in patients with dyslipidemia already on statin therapy.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Dyslipidemia
7. Study Design
Primary Purpose
Treatment
Study Phase
Phase 1
Interventional Study Model
Parallel Assignment
Masking
ParticipantInvestigator
Allocation
Randomized
Enrollment
46 (Actual)
8. Arms, Groups, and Interventions
Arm Title
Panel A
Arm Type
Experimental
Arm Description
Period 1: atorvastatin + placebo to MK0859; Period 2: atorvastatin + MK0859
Arm Title
Panel B
Arm Type
Experimental
Arm Description
Period 1: placebo to atorvastatin + placebo to MK0859; Period 2: MK0859 + placebo to atorvastatin
Intervention Type
Drug
Intervention Name(s)
anacetrapib
Intervention Description
[Intervention Name: MK0859] MK0859 100 mg tablet once daily for 8 weeks.
Intervention Type
Drug
Intervention Name(s)
Comparator: atorvastatin
Intervention Description
Atorvastatin 20 mg tablet once daily for 4 weeks in Period 1 and 8 weeks in Period 2.
Intervention Type
Drug
Intervention Name(s)
Comparator: placebo to MK0859
Intervention Description
Placebo to MK0859 once daily for 4 weeks.
Intervention Type
Drug
Intervention Name(s)
Comparator: placebo to atorvastatin
Intervention Description
Placebo to atorvastatin once daily for 4 weeks in Period 1 and 8 weeks in Period 2.
Primary Outcome Measure Information:
Title
Difference in Production Rate (PR) and Fractional Catabolic Rate (FCR) of Low Density Lipoprotein (LDL) apoB100 following treatment with MK0859 and atorvastatin versus atorvastatin alone
Time Frame
12 weeks
Secondary Outcome Measure Information:
Title
Difference in FCR of LDL apoB100 following treatment with MK0859 versus placebo
Time Frame
12 weeks
10. Eligibility
Sex
All
Minimum Age & Unit of Time
18 Years
Maximum Age & Unit of Time
70 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
Patient's weight has been stable for at least 6 weeks
Patient is in good health based on medical history, physical exam, and laboratory tests
Patient has dyslipidemia
Exclusion Criteria :
Patient has a history of stroke, seizures, or major neurological disorders
Patient has a history of cancer
Patient is currently taking any lipid-lowering medications or substances except for statins
Patient consumes excessive amounts of alcohol or caffeine
Patient has multiple and/or severe allergies to food or drugs
Overall Study Officials:
First Name & Middle Initial & Last Name & Degree
Medical Monitor
Organizational Affiliation
Merck Sharp & Dohme LLC
Official's Role
Study Director
12. IPD Sharing Statement
Citations:
PubMed Identifier
25961461
Citation
Millar JS, Reyes-Soffer G, Jumes P, Dunbar RL, deGoma EM, Baer AL, Karmally W, Donovan DS, Rafeek H, Pollan L, Tohyama J, Johnson-Levonas AO, Wagner JA, Holleran S, Obunike J, Liu Y, Ramakrishnan R, Lassman ME, Gutstein DE, Ginsberg HN, Rader DJ. Anacetrapib lowers LDL by increasing ApoB clearance in mildly hypercholesterolemic subjects. J Clin Invest. 2015 Jun;125(6):2510-22. doi: 10.1172/JCI80025. Epub 2015 May 11. Erratum In: J Clin Invest. 2016 Apr 1;126(4):1603-4.
Results Reference
background
PubMed Identifier
28729361
Citation
Thomas T, Zhou H, Karmally W, Ramakrishnan R, Holleran S, Liu Y, Jumes P, Wagner JA, Hubbard B, Previs SF, Roddy T, Johnson-Levonas AO, Gutstein DE, Marcovina SM, Rader DJ, Ginsberg HN, Millar JS, Reyes-Soffer G. CETP (Cholesteryl Ester Transfer Protein) Inhibition With Anacetrapib Decreases Production of Lipoprotein(a) in Mildly Hypercholesterolemic Subjects. Arterioscler Thromb Vasc Biol. 2017 Sep;37(9):1770-1775. doi: 10.1161/ATVBAHA.117.309549. Epub 2017 Jul 20.
Results Reference
derived
Learn more about this trial
The Effect of MK0859 on Lipoprotein Metabolism in Patients With Dyslipidemia (0859-026 AM3)
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