Multiple Dose Study of TRx0037
Primary Purpose
Alzheimer's Disease
Status
Completed
Phase
Phase 1
Locations
Study Type
Interventional
Intervention
TRx0037
Sponsored by
About this trial
This is an interventional basic science trial for Alzheimer's Disease
Eligibility Criteria
Inclusion Criteria:
- Male and female 55 and over
- No clinically important abnormal physical finding
- No clinically significant lab results
- Normal ECG
- Normal BP and HR
- BMI between 19 and 32
- Weight 50 to 100 kg
- Able to communicate
- Provide written informed consent
- Non smokers
- Males to use contraception
- Females to be surgically sterile or post menopausal
Exclusion Criteria:
- Administration of any IMP other than study drug within 12 weeks before entry
- Use of any prescribed meds, St John's wort, over the counter meds as described in the protocol
- Surgical or medical condition that might interfere with IMP
- History of drug or alcohol abuse
- Clinically significant allergy requiring treatment
- Loss of greater than 400ml of blood within 12 weeks.
- Serious adverse reaction or hypersensitivity to any drug
- Presence of Hep B, Hep c or HIV-1 or HIV-2 at screening
- Presence of G6PD at screening
- History of methaemoglobinaemia
- Partner who is pregnant of lactating
- Positive Pregnancy test
Sites / Locations
Arms of the Study
Arm 1
Arm Type
Experimental
Arm Label
TRx0037
Arm Description
Double blind placebo controlled study of TRx0037 in healthy elderly volunteers to assess safety, tolerability, bioavailability and pharmacokinetics
Outcomes
Primary Outcome Measures
Bioavailability
The bioavailability of TRx0037 in an older population closer to the typical age range of the target patient population.
Pharmacokinetics
The pharmacokinetics for single doses of TRx0037 in healthy elderly volunteers.
Safety and tolerability
Safety and tolerability measurements including adverse events, physical examination findings, vital signs, ECG, and clinical laboratory measurements for single doses of TRx0037
Secondary Outcome Measures
Full Information
NCT ID
NCT01253499
First Posted
December 2, 2010
Last Updated
December 16, 2010
Sponsor
TauRx Therapeutics Ltd
Collaborators
Quotient Clinical
1. Study Identification
Unique Protocol Identification Number
NCT01253499
Brief Title
Multiple Dose Study of TRx0037
Official Title
A Phase 1 Study Consisting of a Double-Blind, Placebo Controlled Multiple Dose Study of TRx0037 in Healthy Elderly Volunteers
Study Type
Interventional
2. Study Status
Record Verification Date
December 2010
Overall Recruitment Status
Completed
Study Start Date
March 2010 (undefined)
Primary Completion Date
May 2010 (Actual)
Study Completion Date
May 2010 (Actual)
3. Sponsor/Collaborators
Name of the Sponsor
TauRx Therapeutics Ltd
Collaborators
Quotient Clinical
4. Oversight
5. Study Description
Brief Summary
The purpose of this study is to evaluate the safety, tolerability and pharmacokinetics of TRx0037 after multiple doses in elderly volunteers.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Alzheimer's Disease
7. Study Design
Primary Purpose
Basic Science
Study Phase
Phase 1
Interventional Study Model
Single Group Assignment
Masking
ParticipantInvestigatorOutcomes Assessor
Allocation
Randomized
Enrollment
31 (Actual)
8. Arms, Groups, and Interventions
Arm Title
TRx0037
Arm Type
Experimental
Arm Description
Double blind placebo controlled study of TRx0037 in healthy elderly volunteers to assess safety, tolerability, bioavailability and pharmacokinetics
Intervention Type
Drug
Intervention Name(s)
TRx0037
Intervention Description
75mg and 100mg tablets used to create doses of 100mg and 175mg. Active placebo 2mg and blank placebo used as comparators.
Primary Outcome Measure Information:
Title
Bioavailability
Description
The bioavailability of TRx0037 in an older population closer to the typical age range of the target patient population.
Time Frame
19 Days (7-10 day follow up)
Title
Pharmacokinetics
Description
The pharmacokinetics for single doses of TRx0037 in healthy elderly volunteers.
Time Frame
19 Days (7-10 day follow up)
Title
Safety and tolerability
Description
Safety and tolerability measurements including adverse events, physical examination findings, vital signs, ECG, and clinical laboratory measurements for single doses of TRx0037
Time Frame
19 Days (7-10 day follow up)
10. Eligibility
Sex
All
Minimum Age & Unit of Time
55 Years
Accepts Healthy Volunteers
Accepts Healthy Volunteers
Eligibility Criteria
Inclusion Criteria:
Male and female 55 and over
No clinically important abnormal physical finding
No clinically significant lab results
Normal ECG
Normal BP and HR
BMI between 19 and 32
Weight 50 to 100 kg
Able to communicate
Provide written informed consent
Non smokers
Males to use contraception
Females to be surgically sterile or post menopausal
Exclusion Criteria:
Administration of any IMP other than study drug within 12 weeks before entry
Use of any prescribed meds, St John's wort, over the counter meds as described in the protocol
Surgical or medical condition that might interfere with IMP
History of drug or alcohol abuse
Clinically significant allergy requiring treatment
Loss of greater than 400ml of blood within 12 weeks.
Serious adverse reaction or hypersensitivity to any drug
Presence of Hep B, Hep c or HIV-1 or HIV-2 at screening
Presence of G6PD at screening
History of methaemoglobinaemia
Partner who is pregnant of lactating
Positive Pregnancy test
Overall Study Officials:
First Name & Middle Initial & Last Name & Degree
Stuart Dr Mair, MBChB
Organizational Affiliation
Quotient Clinical
Official's Role
Principal Investigator
12. IPD Sharing Statement
Learn more about this trial
Multiple Dose Study of TRx0037
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