Safety, Tolerability, Pharmacokinetics and Efficacy of YHD1044
Primary Purpose
Premature Ejaculation
Status
Completed
Phase
Phase 1
Locations
Korea, Republic of
Study Type
Interventional
Intervention
dapoxetine
Sponsored by
About this trial
This is an interventional basic science trial for Premature Ejaculation
Eligibility Criteria
Inclusion Criteria:
- Patient is in a stable, monogamous sexual relationship with the same woman for at least 6 months and plans to maintain this relationship for the duration of the study
- History of premature ejaculation in the 6 months before study initiation
- History of intravaginal ejaculatory latency time (IELT) of < = 2 minutes in at least half of events
- Premature Ejaculation Diagnostic Tool (PEDT) > =11
- 6 domains of International Index of Erectile Function(IIEF) >= 21
- Patient and partner must agree to attempt sexual intercourse at minimum intervals specified in the protocol
- Patient's partner must have a negative urine pregnancy test at time of screening
Exclusion Criteria:
- Medical history which affects ADME in the past 3 years
- Clinically significant and active disorder in ophthalmic system, gastro-intestine, cardiovascular, respiratory system, endocrine system, autoimmune system or malignant tumor,
- Subjects with clinically significant observations considered as unsuitable based on medical judgment in the physical examination and clinical laboratory tests or a medical history
- History of psychological disease
- Clinically significant allergic disease
- Hypersensitivity to TCA, SSRIs(Clomipramine, sertraline, fluoxetine, dapoxetine)
- Taken dapoxetine within 3 months
- Using other forms of therapy for treatment of PE (behavioral therapy or medications applied to the skin)
- Taken another investigational drug within 1 month
- History of drug abuse
Sites / Locations
- Samsung medical center
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm Type
Experimental
Experimental
Experimental
Arm Label
YHD1044 I
YHD1044 III
YHD1044 V
Arm Description
Outcomes
Primary Outcome Measures
Safety and tolerability
through physical examination, laboratory result, vital sign,ECG etc.
Secondary Outcome Measures
Efficacy(IELT)
change from baseline in IELT at the Day 13, 28
Cmax(Cmax,ss), Cmin,ss, AUCinf, AUCt, Tmax, CL/F
Cmax(Cmax,ss), Cmin,ss, AUCinf, AUCt will be assessed. Samping time point: intensive sampling(Day1~2, Day14~15)& intermittent sampling(Day3~Day 28 except intensive sampling period)
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT01419470
Brief Title
Safety, Tolerability, Pharmacokinetics and Efficacy of YHD1044
Official Title
Phase Ⅰ/Ⅱ Clinical Trial to Investigate the Safety, Tolerability, Pharmacokinetics and Efficacy of YHD1044 After Oral Administration in Premature Ejaculation Patients
Study Type
Interventional
2. Study Status
Record Verification Date
July 2012
Overall Recruitment Status
Completed
Study Start Date
February 2011 (undefined)
Primary Completion Date
May 2012 (Actual)
Study Completion Date
May 2012 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Yuhan Corporation
4. Oversight
Data Monitoring Committee
No
5. Study Description
Brief Summary
safety and tolerability, pharmacokinetics/efficacy of an escalating, repeat doses of YHD1044 in premature ejaculation
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Premature Ejaculation
7. Study Design
Primary Purpose
Basic Science
Study Phase
Phase 1, Phase 2
Interventional Study Model
Parallel Assignment
Masking
ParticipantCare ProviderInvestigator
Allocation
Randomized
Enrollment
24 (Actual)
8. Arms, Groups, and Interventions
Arm Title
YHD1044 I
Arm Type
Experimental
Arm Title
YHD1044 III
Arm Type
Experimental
Arm Title
YHD1044 V
Arm Type
Experimental
Intervention Type
Drug
Intervention Name(s)
dapoxetine
Other Intervention Name(s)
Priligy
Intervention Description
multiple dosing
12 subjects will be administered YHD1044 (I, III, V) or active/placebo comparators;dapoxetine
Primary Outcome Measure Information:
Title
Safety and tolerability
Description
through physical examination, laboratory result, vital sign,ECG etc.
Time Frame
throughout the study up to day 28
Secondary Outcome Measure Information:
Title
Efficacy(IELT)
Description
change from baseline in IELT at the Day 13, 28
Time Frame
13days, 28days
Title
Cmax(Cmax,ss), Cmin,ss, AUCinf, AUCt, Tmax, CL/F
Description
Cmax(Cmax,ss), Cmin,ss, AUCinf, AUCt will be assessed. Samping time point: intensive sampling(Day1~2, Day14~15)& intermittent sampling(Day3~Day 28 except intensive sampling period)
Time Frame
specified timepoints in the protocol
10. Eligibility
Sex
Male
Minimum Age & Unit of Time
20 Years
Maximum Age & Unit of Time
60 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
Patient is in a stable, monogamous sexual relationship with the same woman for at least 6 months and plans to maintain this relationship for the duration of the study
History of premature ejaculation in the 6 months before study initiation
History of intravaginal ejaculatory latency time (IELT) of < = 2 minutes in at least half of events
Premature Ejaculation Diagnostic Tool (PEDT) > =11
6 domains of International Index of Erectile Function(IIEF) >= 21
Patient and partner must agree to attempt sexual intercourse at minimum intervals specified in the protocol
Patient's partner must have a negative urine pregnancy test at time of screening
Exclusion Criteria:
Medical history which affects ADME in the past 3 years
Clinically significant and active disorder in ophthalmic system, gastro-intestine, cardiovascular, respiratory system, endocrine system, autoimmune system or malignant tumor,
Subjects with clinically significant observations considered as unsuitable based on medical judgment in the physical examination and clinical laboratory tests or a medical history
History of psychological disease
Clinically significant allergic disease
Hypersensitivity to TCA, SSRIs(Clomipramine, sertraline, fluoxetine, dapoxetine)
Taken dapoxetine within 3 months
Using other forms of therapy for treatment of PE (behavioral therapy or medications applied to the skin)
Taken another investigational drug within 1 month
History of drug abuse
Facility Information:
Facility Name
Samsung medical center
City
Seoul
Country
Korea, Republic of
12. IPD Sharing Statement
Learn more about this trial
Safety, Tolerability, Pharmacokinetics and Efficacy of YHD1044
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