Disulfiram and Chelated Zinc for the Rx of Disseminated Mets Mel That Has Failed First Line Therapy
Primary Purpose
Melanoma
Status
Completed
Phase
Phase 2
Locations
Study Type
Interventional
Intervention
disulfiram and chelated zinc
Sponsored by
About this trial
This is an interventional treatment trial for Melanoma
Eligibility Criteria
Inclusion Criteria:
The subjects must fulfill all the following inclusion criteria to be eligible for participation in the study, unless otherwise specified:
- Male and female patients with stage IV melanoma cancer with biopsy proven metastases demonstrated by imaging studies. Extent of disease should be documented by CT scanning of the chest, abdomen and pelvis, or PET/CT scanning. At least one site of disease should be measurable by RECIST criteria.
- Age of 18 years or more
- ECOG performance status of 0 - 2
- Patients must have received and progressed after or not responded to at least one cycle of first line therapy (chemotherapy, biotherapy, or biochemotherapy) or are unwilling or ineligible to undergo standard therapy
- Patients with brain metastases along with disease at other sites are eligible to participate if their brain disease has been treated with surgery or radiation
- Not currently receiving other cancer chemotherapy
- Not currently participating in another study
- Baseline AST and ALT not greater than 2.0 X upper limit of normal
- Able and willing to provide informed consent and to comply with study procedures
- Able to ingest oral medications
- No known allergy to disulfiram or zinc gluconate
- Willing to refrain from ingestion of alcoholic beverages while on the study
- Serum copper within the normal range at baseline, or if outside the normal range, the PI will review for clinical significance
Exclusion Criteria:
Potential study subjects who meet any of the following criteria are not eligible for participation in the study:
- Participation in another clinical trial of a therapeutic drug during the past 30 days
- Addiction to alcohol or cocaine
- Baseline AST or ALT greater than 2.0 X upper limit of normal
- Unable to ingest oral medications
- Unable to undergo CT scanning because of inability to lie recumbent in the scanner;
- Actively receiving cytotoxic cancer chemotherapy agents
- Evidence of thiuram allergy (may present as contact allergy to rubber or elastic)
- Current use of sertraline and cyclosporine
- Women of child-bearing potential who are not using a commonly accepted effective means of contraception; women of child-bearing potential will have a pregnancy test before enrollment
- Need for warfarin or theophylline, the metabolism of which is likely influenced by disulfiram
- Pregnant women and nursing mothers are not allowed to enroll on this study
- Patients who are taking medications metabolized by cytochrome P450 2E1, including chlorzoxazone or halothane and its derivatives
Sites / Locations
Arms of the Study
Arm 1
Arm Type
Other
Arm Label
Disulfiram and chelated zinc
Arm Description
There is only one arm. All patients are treated wtih disulfiram and chelated zinc.
Outcomes
Primary Outcome Measures
Overall Response Rate to Treatment of Melanoma With Disulfiram and Chelated Zinc
Per Response Evaluation Criteria In Solid Tumors Criteria (RECIST v1.1) for target lesions and assessed by CT scanning of the chest, abdomen and pelvis, or PET/CT scanning.: Complete Response (CR), Disappearance of all target lesions; Partial Response (PR), >=30% decrease in the sum of the longest diameter of target lesions; Overall Response (OR) = CR + PR.
Secondary Outcome Measures
Progression Free Survival
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT02101008
Brief Title
Disulfiram and Chelated Zinc for the Rx of Disseminated Mets Mel That Has Failed First Line Therapy
Study Type
Interventional
2. Study Status
Record Verification Date
December 2015
Overall Recruitment Status
Completed
Study Start Date
March 2010 (undefined)
Primary Completion Date
February 2013 (Actual)
Study Completion Date
undefined (undefined)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
University of Utah
4. Oversight
Data Monitoring Committee
Yes
5. Study Description
Brief Summary
Primary Objectives Determine the response rate associated with treatment of refractory disseminated malignant melanoma with disulfiram and chelated zinc.
Secondary Objectives Determine the progression-free survival associated with treatment of refractory disseminated malignant melanoma with disulfiram and chelated zinc.
Determine the overall survival associated with treatment of refractory disseminated malignant melanoma with disulfiram and chelated zinc.
Determine the toxicity associated with treatment of refractory disseminated malignant melanoma with disulfiram and chelated zinc Determine the effect of disulfiram and chelated zinc on in vivo protein S-glutathionylation.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Melanoma
7. Study Design
Primary Purpose
Treatment
Study Phase
Phase 2
Interventional Study Model
Single Group Assignment
Masking
None (Open Label)
Allocation
N/A
Enrollment
12 (Actual)
8. Arms, Groups, and Interventions
Arm Title
Disulfiram and chelated zinc
Arm Type
Other
Arm Description
There is only one arm. All patients are treated wtih disulfiram and chelated zinc.
Intervention Type
Drug
Intervention Name(s)
disulfiram and chelated zinc
Primary Outcome Measure Information:
Title
Overall Response Rate to Treatment of Melanoma With Disulfiram and Chelated Zinc
Description
Per Response Evaluation Criteria In Solid Tumors Criteria (RECIST v1.1) for target lesions and assessed by CT scanning of the chest, abdomen and pelvis, or PET/CT scanning.: Complete Response (CR), Disappearance of all target lesions; Partial Response (PR), >=30% decrease in the sum of the longest diameter of target lesions; Overall Response (OR) = CR + PR.
Time Frame
Response to treatment will be measured by RECIST evaluation at disease assessment time-points from date of randomization until the date of first documented progression or death from any cause whichever came first (up to five years).
Secondary Outcome Measure Information:
Title
Progression Free Survival
Time Frame
Every 56 days - for up to two years
10. Eligibility
Sex
All
Minimum Age & Unit of Time
18 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
The subjects must fulfill all the following inclusion criteria to be eligible for participation in the study, unless otherwise specified:
Male and female patients with stage IV melanoma cancer with biopsy proven metastases demonstrated by imaging studies. Extent of disease should be documented by CT scanning of the chest, abdomen and pelvis, or PET/CT scanning. At least one site of disease should be measurable by RECIST criteria.
Age of 18 years or more
ECOG performance status of 0 - 2
Patients must have received and progressed after or not responded to at least one cycle of first line therapy (chemotherapy, biotherapy, or biochemotherapy) or are unwilling or ineligible to undergo standard therapy
Patients with brain metastases along with disease at other sites are eligible to participate if their brain disease has been treated with surgery or radiation
Not currently receiving other cancer chemotherapy
Not currently participating in another study
Baseline AST and ALT not greater than 2.0 X upper limit of normal
Able and willing to provide informed consent and to comply with study procedures
Able to ingest oral medications
No known allergy to disulfiram or zinc gluconate
Willing to refrain from ingestion of alcoholic beverages while on the study
Serum copper within the normal range at baseline, or if outside the normal range, the PI will review for clinical significance
Exclusion Criteria:
Potential study subjects who meet any of the following criteria are not eligible for participation in the study:
Participation in another clinical trial of a therapeutic drug during the past 30 days
Addiction to alcohol or cocaine
Baseline AST or ALT greater than 2.0 X upper limit of normal
Unable to ingest oral medications
Unable to undergo CT scanning because of inability to lie recumbent in the scanner;
Actively receiving cytotoxic cancer chemotherapy agents
Evidence of thiuram allergy (may present as contact allergy to rubber or elastic)
Current use of sertraline and cyclosporine
Women of child-bearing potential who are not using a commonly accepted effective means of contraception; women of child-bearing potential will have a pregnancy test before enrollment
Need for warfarin or theophylline, the metabolism of which is likely influenced by disulfiram
Pregnant women and nursing mothers are not allowed to enroll on this study
Patients who are taking medications metabolized by cytochrome P450 2E1, including chlorzoxazone or halothane and its derivatives
12. IPD Sharing Statement
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Disulfiram and Chelated Zinc for the Rx of Disseminated Mets Mel That Has Failed First Line Therapy
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