A Study of Safety, Tolerability, and the Effects Two ND-L02-s0201 Have on the Body
Primary Purpose
Fibrosis
Status
Completed
Phase
Phase 1
Locations
Study Type
Interventional
Intervention
ND-L02-s0201
Sponsored by

About this trial
This is an interventional basic science trial for Fibrosis
Eligibility Criteria
Inclusion Criteria:
- Subject is in good health, as determined by the Investigator
- Subject consumes an average of no more than 2 alcoholic drinks per day within the 6 months before administration of study drug
- Subject has serum calcium and parathyroid hormone (intact) within the limits of the normal range of the laboratory
Exclusion Criteria:
- Subject has a disease or condition (medical or surgical) which, in the opinion of the Investigator, may compromise the hematologic, cardiovascular, pulmonary, renal, gastrointestinal, hepatic, skeletal, or central nervous systems; or other conditions that may interfere with the absorption, distribution, metabolism, or excretion of ND-L02-s0201 solution, or that may place the subject at increased risk
- Subject has a history of bone disease, including osteoporosis and osteomalacia, Paget's disease of bone, or a history of unexplained fractures or fractures after minimal trauma
- Subject has abnormal laboratory values considered to be clinically significant by the Investigator
Other protocol inclusion/exclusion criteria may apply
Sites / Locations
Arms of the Study
Arm 1
Arm 2
Arm Type
Experimental
Experimental
Arm Label
Module A
Module B
Arm Description
Lyophilized Formulation
Frozen Formulation
Outcomes
Primary Outcome Measures
Maximum plasma concentration (Cmax)
Time to maximum plasma concentration (Tmax)
Area under the plasma concentration-time curve from time 0 to the last available observable concentration (AUC0-t)
Area under the plasma concentration-time curve extrapolated to infinity (AUC0-∞)
Area under the first moment of the plasma concentration-time curve from time zero to infinity (AUMC0-inf)
Apparent first-order terminal elimination rate constant (Kel)
Volume of distribution during the elimination phase after IV administration (Vz)
Apparent volume of distribution at steady-state (Vss)
Total plasma clearance of drug after IV administration (CL/F)
Apparent first-order terminal elimination half-life (T1/2)
Secondary Outcome Measures
Incidence of adverse events (AEs)
Incidence of serious adverse events (SAEs)
Incidence of discontinuations of study drug due to toxicity
Full Information
NCT ID
NCT03241264
First Posted
August 3, 2017
Last Updated
August 3, 2017
Sponsor
Bristol-Myers Squibb
Collaborators
Nitto Denko Corporation
1. Study Identification
Unique Protocol Identification Number
NCT03241264
Brief Title
A Study of Safety, Tolerability, and the Effects Two ND-L02-s0201 Have on the Body
Official Title
A Phase 1, Open-Label, Randomized-Sequence, Single-Crossover, Bridging Study to Evaluate the Single-Dose Pharmacokinetics, Safety, and Tolerability of Two ND-L02-s0201 Formulations, Frozen Versus Lyophilized, Administered by Intravenous Infusion to Healthy Male and Female Subjects
Study Type
Interventional
2. Study Status
Record Verification Date
July 2017
Overall Recruitment Status
Completed
Study Start Date
August 28, 2016 (Actual)
Primary Completion Date
October 21, 2016 (Actual)
Study Completion Date
October 21, 2016 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Bristol-Myers Squibb
Collaborators
Nitto Denko Corporation
4. Oversight
Studies a U.S. FDA-regulated Drug Product
Yes
Studies a U.S. FDA-regulated Device Product
No
Data Monitoring Committee
No
5. Study Description
Brief Summary
The purpose of this study is to evaluate the safety, tolerability, and the effects two ND-L02-s0201 have on the body
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Fibrosis
7. Study Design
Primary Purpose
Basic Science
Study Phase
Phase 1
Interventional Study Model
Crossover Assignment
Masking
None (Open Label)
Allocation
Randomized
Enrollment
12 (Actual)
8. Arms, Groups, and Interventions
Arm Title
Module A
Arm Type
Experimental
Arm Description
Lyophilized Formulation
Arm Title
Module B
Arm Type
Experimental
Arm Description
Frozen Formulation
Intervention Type
Drug
Intervention Name(s)
ND-L02-s0201
Intervention Description
Specified dose on specified day
Primary Outcome Measure Information:
Title
Maximum plasma concentration (Cmax)
Time Frame
Up to 28 days
Title
Time to maximum plasma concentration (Tmax)
Time Frame
Up to 28 days
Title
Area under the plasma concentration-time curve from time 0 to the last available observable concentration (AUC0-t)
Time Frame
Up to 28 days
Title
Area under the plasma concentration-time curve extrapolated to infinity (AUC0-∞)
Time Frame
Up to 28 days
Title
Area under the first moment of the plasma concentration-time curve from time zero to infinity (AUMC0-inf)
Time Frame
Up to 28 days
Title
Apparent first-order terminal elimination rate constant (Kel)
Time Frame
Up to 28 days
Title
Volume of distribution during the elimination phase after IV administration (Vz)
Time Frame
Up to 28 days
Title
Apparent volume of distribution at steady-state (Vss)
Time Frame
Up to 28 days
Title
Total plasma clearance of drug after IV administration (CL/F)
Time Frame
Up to 28 days
Title
Apparent first-order terminal elimination half-life (T1/2)
Time Frame
Up to 28 days
Secondary Outcome Measure Information:
Title
Incidence of adverse events (AEs)
Time Frame
Up to 28 days
Title
Incidence of serious adverse events (SAEs)
Time Frame
Up to 28 days
Title
Incidence of discontinuations of study drug due to toxicity
Time Frame
Up to 28 days
10. Eligibility
Sex
All
Minimum Age & Unit of Time
18 Years
Maximum Age & Unit of Time
55 Years
Accepts Healthy Volunteers
Accepts Healthy Volunteers
Eligibility Criteria
Inclusion Criteria:
Subject is in good health, as determined by the Investigator
Subject consumes an average of no more than 2 alcoholic drinks per day within the 6 months before administration of study drug
Subject has serum calcium and parathyroid hormone (intact) within the limits of the normal range of the laboratory
Exclusion Criteria:
Subject has a disease or condition (medical or surgical) which, in the opinion of the Investigator, may compromise the hematologic, cardiovascular, pulmonary, renal, gastrointestinal, hepatic, skeletal, or central nervous systems; or other conditions that may interfere with the absorption, distribution, metabolism, or excretion of ND-L02-s0201 solution, or that may place the subject at increased risk
Subject has a history of bone disease, including osteoporosis and osteomalacia, Paget's disease of bone, or a history of unexplained fractures or fractures after minimal trauma
Subject has abnormal laboratory values considered to be clinically significant by the Investigator
Other protocol inclusion/exclusion criteria may apply
12. IPD Sharing Statement
Learn more about this trial
A Study of Safety, Tolerability, and the Effects Two ND-L02-s0201 Have on the Body
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