A Study to Evaluate the Safety, Pharmacokinetics, and Activity of GDC-6036 Alone or in Combination in Participants With Advanced or Metastatic Solid Tumors With a KRAS G12C Mutation
Non-Small Cell Lung Cancer, Colorectal Cancer, Advanced Solid Tumors
About this trial
This is an interventional treatment trial for Non-Small Cell Lung Cancer focused on measuring KRAS G12C, Non-Small Cell Lung Cancer, Colorectal Cancer, GDC-6036, Metastatic Solid Tumor, Atezolizumab, Bevacizumab, Cetuximab, Erlotinib, Inavolisib, GDC-1971, SHP2
Eligibility Criteria
Inclusion Criteria:
- Histologically documented advanced or metastatic solid tumor with KRAS G12C mutation.
- Women of childbearing potential must agree to remain abstinent or use contraception, and agree to refrain from donating eggs during the treatment period and after the final dose of study treatment as specified in the protocol.
- Men who are not surgically sterile must agree to remain abstinent or use a condom, and agreement to refrain from donating sperm during the treatment period and after the final dose of study treatment as specified in the protocol.
Exclusion Criteria:
- Active brain metastases.
- Malabsorption or other condition that interferes with enteral absorption.
- Clinically significant cardiovascular dysfunction or liver disease.
Sites / Locations
- City of Hope Comprehensive Cancer CenterRecruiting
- UCSD Moores Cancer CenterRecruiting
- Chao Family Comprehensive Cancer Center UCIRecruiting
- Univ of Calif, San Francisco; Breast Cancer CenterRecruiting
- Yale Cancer CenterRecruiting
- Florida Cancer Specialists - SarasotaRecruiting
- Dana Farber Cancer InstituteRecruiting
- Memorial Sloan Kettering Cancer CenterRecruiting
- University of Oklahoma; Stephenson Oklahoma Canc CtrRecruiting
- Abramson Cancer Center; Univ of PennsylvaniaRecruiting
- UPMC - Hillman Cancer CenterRecruiting
- St Vincent's Hospital SydneyRecruiting
- Slade Health Inward goodsRecruiting
- Alfred HealthRecruiting
- Peter MacCallum Cancer CenterRecruiting
- Linear Clinical Research LimitedRecruiting
- UZ AntwerpenRecruiting
- CHU de LiègeRecruiting
- AZ St Maarten Campus LeopoldstrRecruiting
- Santa Casa de Misericórdia de Belo Horizonte - PPDSRecruiting
- Hospital de Clinicas de Porto Alegre HCPA PPDSRecruiting
- Hospital Erasto GaertnerRecruiting
- Instituto Nacional de CâncerRecruiting
- Universidade de Caxias do SulRecruiting
- Hospital Sao Lucas Da Pontificia Universidade Catolica Do Rio Grande Do Sul (PUCRS)Recruiting
- Hospital de Cancer de BarretosRecruiting
- Fundacao Faculdade Regional de Medicina de Sao Jose Do Rio Preto Hospital de Base - PPDSRecruiting
- Instituto do Cancer do Estado de Sao Paulo - ICESPRecruiting
- Ottawa HospitalRecruiting
- Princess Margaret Cancer CentreRecruiting
- Jewish General Hospital; Sir Mortimer B. DavisRecruiting
- Semmelweis EgyetemRecruiting
- Clinexpert Kft. - GyongyosRecruiting
- Rambam Medical CenterRecruiting
- Sheba Medical Center - PPDSRecruiting
- Tel-Aviv Sourasky Medical CenterRecruiting
- Istituto Scientifico Romagnolo Per Lo Studio E La Cura Dei Tumori IRST - PPDS
- Irccs Ospedale San Raffaele;Oncologia MedicaRecruiting
- Asst Grande Ospedale Metropolitano NiguardaRecruiting
- Istituto Clinico HumanitasRecruiting
- Azienda Ospedaliero Universitaria PisanaRecruiting
- Aga Khan University HospitalRecruiting
- Seoul National University Bundang HospitalRecruiting
- Seoul National University HospitalRecruiting
- Asan Medical Center - PPDSRecruiting
- Samsung Medical Center - PPDSRecruiting
- Het Nederlands Kanker Instituut Antoni Van Leeuwenhoek ZiekenhuisRecruiting
- Leids Universitair Medisch CentrumRecruiting
- Maastricht University Medical CenterRecruiting
- Universitair Medisch Centrum UtrechtRecruiting
- Auckland City Hospital, Cancer and Blood ResearchRecruiting
- Auckland City HospitalRecruiting
- New Zealand Clinical Research - ChristchurchRecruiting
- Haukeland University Hospital; Hospital PharmacyRecruiting
- Oslo university hospital RadiumhospitaletRecruiting
- Medical University of GdanskRecruiting
- Biokinetica, Przychodnia JozefowRecruiting
- Uniwersytecki Szpital Kliniczny w PoznaniuRecruiting
- Republican Clinical Oncology Dispensary of Ministry of Healthcare of Tatarstan Republic
- Hospital Universitari Vall d'HebronRecruiting
- START Madrid-FJD, Hospital Fundacion Jimenez DiazRecruiting
- Hospital Universitario 12 de OctubreRecruiting
- Hospital Universitario HM Sanchinarro-CIOCCRecruiting
- Hospital Clinico Universitario Virgen de la VictoriaRecruiting
- Hospital Universitario Virgen del RocíoRecruiting
- Hospital Clinico Universitario de ValenciaRecruiting
- Universitaetsspital Basel; Onkologie
- InselspitalRecruiting
- Hôpitaux Universitaires de GenèveRecruiting
- Unversitätsspital Zürich
- Queen Elizabeth HospitalRecruiting
- Velindre Cancer CentreRecruiting
- University College London Hospitals NHS Foundation Trust; NIHR UCLH Clinical Research FacilityRecruiting
- The Christie NHS Foundation TrustRecruiting
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm 4
Arm 5
Arm 6
Arm 7
Experimental
Experimental
Experimental
Experimental
Experimental
Experimental
Experimental
Arm A: Dose-escalation (Stage I), Dose Expansion (Stage II)
Arm B: GDC-6036 + Atezolizumab (Stage I and Stage II)
Arm C: GDC-6036 + Cetuximab (Stage I and Stage II)
Arm D: GDC-6036 + Bevacizumab (Stage I and Stage II)
Arm E: GDC-6036 + Erlotinib (Stage I and Stage II)
Arm F: GDC-6036 + GDC-1971 (Stage I and Stage II)
Arm G: GDC-6036 + Inavolisib (Stage I and Stage II)
Participants in Stage I will receive GDC-6036 administered orally once daily (PO QD). The dose will be increased in successive cohorts until a study-specific threshold is reached. Participants with select solid tumors will be treated with GDC-6036 PO QD in Stage II.
Participants with non-small cell lung cancer will receive GDC-6036 in combination with atezolizumab.
Participants with colorectal cancer will receive GDC-6036 in combination with cetuximab.
Participants with solid tumors will receive GDC-6036 in combination with bevacizumab.
Participants with non-small cell lung cancer will receive GDC-6036 in combination with erlotinib.
Participants with solid tumors will receive GDC-6036 in combination with GDC-1971 PO in Stage I. Participants with select solid tumors will be treated with GDC-6036 in combination with GDC-1971 PO in Stage II.
Participants with solid tumors will receive GDC-6036 in combination with inavolisib PO in Stage I. Participants with select solid tumors will be treated with GDC-6036 in combination with inavolisib PO in Stage II.