An Exploratory PET-study of Deposition, Disposition and Brain Uptake of [11C]Nicotine After Inhalation of 2 Nicotine Formulations Via the myBluTM E-cigarette in Smokers
Primary Purpose
Healthy Volunteers
Status
Completed
Phase
Not Applicable
Locations
Sweden
Study Type
Interventional
Intervention
myBluTM Formulation 1
myBluTM Formulation 2
Sponsored by
About this trial
This is an interventional other trial for Healthy Volunteers
Eligibility Criteria
Inclusion Criteria:
- Body mass index ≥18.0 and ≤ 30.0 kg/m2
- Habitual daily cigarette smoker
- Women have to be of non-child bearing potential
Exclusion Criteria:
- History of any clinically significant disease
- Relevant concomitant medication
- Any clinically significant condition
- Malignancy within the past 5 years
- Positif for HIV, hepatitis B or C
- Untreated hypertension
- Previous participation to a PET-study or other nuclide medical study
- Previous exposure to significant radiation
- Negative results of the modified Allen test on both arms at screening
- Alcohol or drug abuse
Sites / Locations
- PET Centre, Uppsala University Hospital
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm 4
Arm Type
Experimental
Experimental
Experimental
Experimental
Arm Label
myBluTM Formulation 1 Oral cavity and lungs
myBluTM Formulation 2 Oral cavity and lungs
myBluTM Formulation 1 Brain
myBluTM Formulation 2 Brain
Arm Description
This group was used for measuring oral cavity and lungs endpoints after administration of Formulation 1
This group was used for measuring oral cavity and lungs endpoints after administration of Formulation 2
This group was used for measuring brain endpoints after administration of Formulation 1
This group was used for measuring brain endpoints after administration of Formulation 2
Outcomes
Primary Outcome Measures
Lung PET
Peak accumulation of [11C]nicotine deposited in the lung during 40 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the lungs
Oral Cavity PET
Peak accumulation of nicotine deposited in the oral cavity during 40 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the oral cavity
Brain PET
Peak accumulation of nicotine deposited in the brain during 30 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the brain
Secondary Outcome Measures
Full Information
NCT ID
NCT04780815
First Posted
February 23, 2021
Last Updated
July 8, 2022
Sponsor
Imperial Brands PLC
Collaborators
Nerudia Ltd
1. Study Identification
Unique Protocol Identification Number
NCT04780815
Brief Title
An Exploratory PET-study of Deposition, Disposition and Brain Uptake of [11C]Nicotine After Inhalation of 2 Nicotine Formulations Via the myBluTM E-cigarette in Smokers
Official Title
An Exploratory PET-study of Deposition, Disposition and Brain Uptake of [11C]Nicotine After Inhalation of 2 Nicotine Formulations Via the myBluTM E-cigarette in Smokers
Study Type
Interventional
2. Study Status
Record Verification Date
July 2022
Overall Recruitment Status
Completed
Study Start Date
March 16, 2020 (Actual)
Primary Completion Date
November 17, 2020 (Actual)
Study Completion Date
November 17, 2020 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Imperial Brands PLC
Collaborators
Nerudia Ltd
4. Oversight
Studies a U.S. FDA-regulated Drug Product
No
Studies a U.S. FDA-regulated Device Product
No
5. Study Description
Brief Summary
This is a single-center, exploratory positron emission tomography (PET) study of deposition, disposition and brain uptake [11C]nicotine when given to smokers as two different formulations via mybluTM e-cigarette system.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Healthy Volunteers
7. Study Design
Primary Purpose
Other
Study Phase
Not Applicable
Interventional Study Model
Parallel Assignment
Masking
None (Open Label)
Allocation
Non-Randomized
Enrollment
16 (Actual)
8. Arms, Groups, and Interventions
Arm Title
myBluTM Formulation 1 Oral cavity and lungs
Arm Type
Experimental
Arm Description
This group was used for measuring oral cavity and lungs endpoints after administration of Formulation 1
Arm Title
myBluTM Formulation 2 Oral cavity and lungs
Arm Type
Experimental
Arm Description
This group was used for measuring oral cavity and lungs endpoints after administration of Formulation 2
Arm Title
myBluTM Formulation 1 Brain
Arm Type
Experimental
Arm Description
This group was used for measuring brain endpoints after administration of Formulation 1
Arm Title
myBluTM Formulation 2 Brain
Arm Type
Experimental
Arm Description
This group was used for measuring brain endpoints after administration of Formulation 2
Intervention Type
Other
Intervention Name(s)
myBluTM Formulation 1
Intervention Description
1-2 puffs of each 3-5 seconds duration taken from myBluTM with Formulation 1, with inhalation of the vapour into the lungs
Intervention Type
Other
Intervention Name(s)
myBluTM Formulation 2
Intervention Description
1-2 puffs of each 3-5 seconds duration taken from myBluTM with Formulation 2, with inhalation of the vapour into the lungs
Primary Outcome Measure Information:
Title
Lung PET
Description
Peak accumulation of [11C]nicotine deposited in the lung during 40 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the lungs
Time Frame
40 minutes
Title
Oral Cavity PET
Description
Peak accumulation of nicotine deposited in the oral cavity during 40 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the oral cavity
Time Frame
40 minutes
Title
Brain PET
Description
Peak accumulation of nicotine deposited in the brain during 30 minutes after product administration, using dynamic PET Digital Imaging and Communications in Medicine (DICOM) images over the brain
Time Frame
30 minutes
10. Eligibility
Sex
All
Minimum Age & Unit of Time
50 Years
Maximum Age & Unit of Time
65 Years
Accepts Healthy Volunteers
Accepts Healthy Volunteers
Eligibility Criteria
Inclusion Criteria:
Body mass index ≥18.0 and ≤ 30.0 kg/m2
Habitual daily cigarette smoker
Women have to be of non-child bearing potential
Exclusion Criteria:
History of any clinically significant disease
Relevant concomitant medication
Any clinically significant condition
Malignancy within the past 5 years
Positif for HIV, hepatitis B or C
Untreated hypertension
Previous participation to a PET-study or other nuclide medical study
Previous exposure to significant radiation
Negative results of the modified Allen test on both arms at screening
Alcohol or drug abuse
Facility Information:
Facility Name
PET Centre, Uppsala University Hospital
City
Uppsala
ZIP/Postal Code
SE-751 85
Country
Sweden
12. IPD Sharing Statement
Plan to Share IPD
No
Learn more about this trial
An Exploratory PET-study of Deposition, Disposition and Brain Uptake of [11C]Nicotine After Inhalation of 2 Nicotine Formulations Via the myBluTM E-cigarette in Smokers
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