A Dose-Finding Study in Japanese Patients to Evaluate the Effect of Obicetrapib as an Adjunct to Stable Statin Therapy.
Primary Purpose
Dyslipidemia, Hypercholesterolemia, High Cholesterol
Status
Completed
Phase
Phase 2
Locations
Japan
Study Type
Interventional
Intervention
Obicetrapib
Obicetrapib
Sponsored by
About this trial
This is an interventional treatment trial for Dyslipidemia focused on measuring obicetrapib, statin, LDL-C cholestero, l atherosclerosis
Eligibility Criteria
Inclusion Criteria:
- LDL-C > 70 mg/dL and TG < 400 mg/dL,
- Treated with a stable statin therapy; Atorvastatin 20/40 or Simvastatin 10/20
Exclusion Criteria:
- BMI > or =35 kg/m2
- Significant cardiovascular disease
- HbA1c > 10%
- Uncontrolled hypertension
- Active muscle disease
- GFR < 60 ml/min
- Hepatic dysfunction
- Anemia
- Existing CETP deficiency
- History of Homozygous Familial Hypercholerstrolemia
- History of malignancy
- Alcohol abuse
- Treatment with investigational product
- Treatment with PCSK9
- Clinically significant condition
- Known CETP inhibitor allergy
Sites / Locations
- Nippon Kokan Fukuyama Hospital
- Nakamura Cardiology and Cardiovascular Surgery Clinic
- Kishiwada Tokushu-Kai Hospital
- Kyosokai AMC NISHI-UMEDA Clinic
- Sakurabashi Watanabe Hospital
- Uji Tokushu-Kai Hospital
- Sanai Hospital
- Shinden Higashi Clinic
- Soka-Sugiura Clinic
- Sugiura Clinic
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm 4
Arm Type
Placebo Comparator
Experimental
Experimental
Experimental
Arm Label
Placebo
Experimental 2.5 mg Obicetrapib
Experimental 5 mg Obicetrapib
Experimental 10 mg Obicetrapib
Arm Description
Once-daily placebo
once-daily Obicetrapib
once-daily Obicetrapib
once-daily Obicetrapib
Outcomes
Primary Outcome Measures
LDL-C
percent change in LDL-C
Secondary Outcome Measures
Apo B
percent change in Apo B
Non-HDL-C
percent change in Non-HDL-C
HDL-C
percent change in HDL-C
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT05421078
Brief Title
A Dose-Finding Study in Japanese Patients to Evaluate the Effect of Obicetrapib as an Adjunct to Stable Statin Therapy.
Official Title
A Placebo-Controlled, Double-Blind, Randomized, Phase 2 Dose-Finding Study to Evaluate the Effect of Obicetrapib as an Adjunct to Stable Statin Therapy in Japanese Subjects.
Study Type
Interventional
2. Study Status
Record Verification Date
July 2023
Overall Recruitment Status
Completed
Study Start Date
June 27, 2022 (Actual)
Primary Completion Date
April 21, 2023 (Actual)
Study Completion Date
August 23, 2023 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
NewAmsterdam Pharma
4. Oversight
Studies a U.S. FDA-regulated Drug Product
Yes
Studies a U.S. FDA-regulated Device Product
No
Product Manufactured in and Exported from the U.S.
Yes
Data Monitoring Committee
No
5. Study Description
Brief Summary
This study will be a placebo-controlled, double-blind, randomized, phase 2 dose-finding study in Japanese patients to evaluate the efficacy, safety, and tolerability of obicetrapib as an adjunct to stable statin therapy.
Detailed Description
This study will be a placebo-controlled, double-blind, randomized, phase 2 dose-finding study to evaluate the efficacy, safety, and tolerability of obicetrapib as an adjunct to stable statin therapy in Japanese patients. The screening period for this study will take up to 2-weeks. Afterwards, patients will be randomized to placebo, 2.5 mg obicetrapib, 5 mg obicetrapib or 10 mg obicetrapib for an 8-week treatment period. After the treatment period, patients will continue for a 4-week safety follow-up visit.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Dyslipidemia, Hypercholesterolemia, High Cholesterol
Keywords
obicetrapib, statin, LDL-C cholestero, l atherosclerosis
7. Study Design
Primary Purpose
Treatment
Study Phase
Phase 2
Interventional Study Model
Parallel Assignment
Model Description
Placebo-controlled, double-blind, randomized
Masking
ParticipantCare ProviderInvestigatorOutcomes Assessor
Masking Description
placebo tablet made to resemble active product
Allocation
Randomized
Enrollment
108 (Actual)
8. Arms, Groups, and Interventions
Arm Title
Placebo
Arm Type
Placebo Comparator
Arm Description
Once-daily placebo
Arm Title
Experimental 2.5 mg Obicetrapib
Arm Type
Experimental
Arm Description
once-daily Obicetrapib
Arm Title
Experimental 5 mg Obicetrapib
Arm Type
Experimental
Arm Description
once-daily Obicetrapib
Arm Title
Experimental 10 mg Obicetrapib
Arm Type
Experimental
Arm Description
once-daily Obicetrapib
Intervention Type
Drug
Intervention Name(s)
Obicetrapib
Other Intervention Name(s)
CETP inhibitor
Intervention Description
tablet
Intervention Type
Drug
Intervention Name(s)
Obicetrapib
Other Intervention Name(s)
placebo tablet
Intervention Description
No active ingredient
Primary Outcome Measure Information:
Title
LDL-C
Description
percent change in LDL-C
Time Frame
8 weeks
Secondary Outcome Measure Information:
Title
Apo B
Description
percent change in Apo B
Time Frame
8 weeks
Title
Non-HDL-C
Description
percent change in Non-HDL-C
Time Frame
8 weeks
Title
HDL-C
Description
percent change in HDL-C
Time Frame
8 weeks
10. Eligibility
Sex
All
Minimum Age & Unit of Time
18 Years
Maximum Age & Unit of Time
75 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
LDL-C > 70 mg/dL and TG < 400 mg/dL,
Treated with a stable statin therapy; Atorvastatin 20/40 or Simvastatin 10/20
Exclusion Criteria:
BMI > or =35 kg/m2
Significant cardiovascular disease
HbA1c > 10%
Uncontrolled hypertension
Active muscle disease
GFR < 60 ml/min
Hepatic dysfunction
Anemia
Existing CETP deficiency
History of Homozygous Familial Hypercholerstrolemia
History of malignancy
Alcohol abuse
Treatment with investigational product
Treatment with PCSK9
Clinically significant condition
Known CETP inhibitor allergy
Overall Study Officials:
First Name & Middle Initial & Last Name & Degree
Marc Ditmarsch, MD
Organizational Affiliation
NewAmsterdam Pharma
Official's Role
Study Director
Facility Information:
Facility Name
Nippon Kokan Fukuyama Hospital
City
Fukuyama
Country
Japan
Facility Name
Nakamura Cardiology and Cardiovascular Surgery Clinic
City
Itoshima
Country
Japan
Facility Name
Kishiwada Tokushu-Kai Hospital
City
Osaka
Country
Japan
Facility Name
Kyosokai AMC NISHI-UMEDA Clinic
City
Osaka
Country
Japan
Facility Name
Sakurabashi Watanabe Hospital
City
Osaka
Country
Japan
Facility Name
Uji Tokushu-Kai Hospital
City
Osaka
Country
Japan
Facility Name
Sanai Hospital
City
Saitama
Country
Japan
Facility Name
Shinden Higashi Clinic
City
Sendai
Country
Japan
Facility Name
Soka-Sugiura Clinic
City
Soka
Country
Japan
Facility Name
Sugiura Clinic
City
Tokyo
Country
Japan
12. IPD Sharing Statement
Plan to Share IPD
No
Learn more about this trial
A Dose-Finding Study in Japanese Patients to Evaluate the Effect of Obicetrapib as an Adjunct to Stable Statin Therapy.
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