Impact of THN102 on Attention, Wakefulness and Cognitive Performance During Total Sleep Deprivation
Primary Purpose
Sleep Deprivation
Status
Completed
Phase
Phase 1
Locations
Study Type
Interventional
Intervention
Placebo
Modafinil
THN102
Sponsored by
About this trial
This is an interventional treatment trial for Sleep Deprivation focused on measuring modafinil, connexin, sleep deprivation, cognitive performance
Eligibility Criteria
Main inclusion Criteria:
- Male subjects considered healthy and aged between 18 and 40 years
- Subject with a body mass index (BMI) between 18 and 30 kg/m2
Sites / Locations
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm 4
Arm 5
Arm Type
Placebo Comparator
Active Comparator
Experimental
Experimental
Experimental
Arm Label
PBO
MOD
THN102 100/1
THN102 100/3
THN102 100/9
Arm Description
Placebo
Modafinil 100mg
modafinil 100 mg + 1 mg flecainide
modafinil 100 mg + 3 mg flecainide
modafinil 100 mg + 9 mg flecainide
Outcomes
Primary Outcome Measures
Sustained attention (PVT)
Mean speed at the 10 min Psychomotor vigilance test (PVT)
Secondary Outcome Measures
Sustained attention (PVT) AUC
AUC of speed values at the 10 min Psychomotor vigilance test (PVT)
Mental flexibility
Wisconsin card sorting test
Mental inhibition
GO-noGO
Working memory
2-Back
Full Information
NCT ID
NCT03182413
First Posted
June 6, 2017
Last Updated
June 8, 2017
Sponsor
Theranexus
Collaborators
Institut de recherche biomédicale des armées (IRBA), Bretigny sur Orge, France
1. Study Identification
Unique Protocol Identification Number
NCT03182413
Brief Title
Impact of THN102 on Attention, Wakefulness and Cognitive Performance During Total Sleep Deprivation
Official Title
Therapeutic Impact of THN102 on Attention, Wakefulness and Cognitive Performance During Total Sleep Deprivation in Healthy Subjects
Study Type
Interventional
2. Study Status
Record Verification Date
June 2017
Overall Recruitment Status
Completed
Study Start Date
September 2015 (undefined)
Primary Completion Date
December 2015 (Actual)
Study Completion Date
March 2016 (Actual)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Theranexus
Collaborators
Institut de recherche biomédicale des armées (IRBA), Bretigny sur Orge, France
4. Oversight
Data Monitoring Committee
Yes
5. Study Description
Brief Summary
Study Objectives: THN102 is a new combination between modafinil and flecainide low-dose, a documented glial connexin inhibitor. Efficacy of THN102 was compared to modafinil and to placebo on parameters impaired by total sleep deprivation (SD, lasting 40h).
Methods: 20 healthy male subjects participated in a double-blind, randomised, incomplete-block 3-period cross-over trial involving 5 treatments (n=12 per group): placebo (PBO), modafinil 100 mg (MOD), and combinations THN102 (modafinil 100 mg and 1, 3 or 9 mg flecainide as THN1, THN3 and THN9), as 3 oral doses over 18h.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Sleep Deprivation
Keywords
modafinil, connexin, sleep deprivation, cognitive performance
7. Study Design
Primary Purpose
Treatment
Study Phase
Phase 1
Interventional Study Model
Crossover Assignment
Masking
ParticipantCare ProviderInvestigatorOutcomes Assessor
Allocation
Randomized
Enrollment
20 (Actual)
8. Arms, Groups, and Interventions
Arm Title
PBO
Arm Type
Placebo Comparator
Arm Description
Placebo
Arm Title
MOD
Arm Type
Active Comparator
Arm Description
Modafinil 100mg
Arm Title
THN102 100/1
Arm Type
Experimental
Arm Description
modafinil 100 mg + 1 mg flecainide
Arm Title
THN102 100/3
Arm Type
Experimental
Arm Description
modafinil 100 mg + 3 mg flecainide
Arm Title
THN102 100/9
Arm Type
Experimental
Arm Description
modafinil 100 mg + 9 mg flecainide
Intervention Type
Drug
Intervention Name(s)
Placebo
Intervention Type
Drug
Intervention Name(s)
Modafinil
Intervention Type
Drug
Intervention Name(s)
THN102
Primary Outcome Measure Information:
Title
Sustained attention (PVT)
Description
Mean speed at the 10 min Psychomotor vigilance test (PVT)
Time Frame
5 hours post treatment
Secondary Outcome Measure Information:
Title
Sustained attention (PVT) AUC
Description
AUC of speed values at the 10 min Psychomotor vigilance test (PVT)
Time Frame
AUC of PVT speed during TSD
Title
Mental flexibility
Description
Wisconsin card sorting test
Time Frame
16,5 hours post treatment
Title
Mental inhibition
Description
GO-noGO
Time Frame
16,5 hours post treatment
Title
Working memory
Description
2-Back
Time Frame
16,5 hours post treatment
10. Eligibility
Sex
Male
Minimum Age & Unit of Time
18 Years
Maximum Age & Unit of Time
40 Years
Accepts Healthy Volunteers
Accepts Healthy Volunteers
Eligibility Criteria
Main inclusion Criteria:
Male subjects considered healthy and aged between 18 and 40 years
Subject with a body mass index (BMI) between 18 and 30 kg/m2
Overall Study Officials:
First Name & Middle Initial & Last Name & Degree
Fabien Sauvet, MD, PhD
Organizational Affiliation
Institut de Recherche Biomedicale des Armees
Official's Role
Principal Investigator
First Name & Middle Initial & Last Name & Degree
Françoise Brunner-Ferber, PhD
Organizational Affiliation
Brunner Naga
Official's Role
Study Director
12. IPD Sharing Statement
Plan to Share IPD
Undecided
Citations:
PubMed Identifier
27091533
Citation
Duchene A, Perier M, Zhao Y, Liu X, Thomasson J, Chauveau F, Pierard C, Lagarde D, Picoli C, Jeanson T, Mouthon F, Dauvilliers Y, Giaume C, Lin JS, Charveriat M. Impact of Astroglial Connexins on Modafinil Pharmacological Properties. Sleep. 2016 Jun 1;39(6):1283-92. doi: 10.5665/sleep.5854.
Results Reference
background
PubMed Identifier
31419329
Citation
Sauvet F, Erblang M, Gomez-Merino D, Rabat A, Guillard M, Dubourdieu D, Lefloch H, Drogou C, Van Beers P, Bougard C, Bourrrilhon C, Arnal P, Rein W, Mouthon F, Brunner-Ferber F, Leger D, Dauvilliers Y, Chennaoui M, Charveriat M. Efficacy of THN102 (a combination of modafinil and flecainide) on vigilance and cognition during 40-hour total sleep deprivation in healthy subjects: Glial connexins as a therapeutic target. Br J Clin Pharmacol. 2019 Nov;85(11):2623-2633. doi: 10.1111/bcp.14098. Epub 2019 Sep 15.
Results Reference
derived
Links:
URL
http://www.theranexus.com
Description
Related Info
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Impact of THN102 on Attention, Wakefulness and Cognitive Performance During Total Sleep Deprivation
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