Oral Axl/Mer/CSF1R Selective Tyrosine Kinase Inhibitor in Patients With Advanced Solid Tumor
Primary Purpose
Solid Tumor, Advanced Cancer, Metastatic Cancer
Status
Recruiting
Phase
Phase 1
Locations
United States
Study Type
Interventional
Intervention
Q702
Sponsored by
About this trial
This is an interventional treatment trial for Solid Tumor
Eligibility Criteria
Inclusion Criteria:
- Patients with histologically or cytologically confirmed advanced or metastatic solid tumors, that have progressed following standard of care therapy or for which there is no standard therapy which confers clinical benefit
- Measurable disease per RECIST v 1.1
- ECOG performance status 0 or 1
- Life expectancy of at least 3 months
- Age ≥ 18 years
- Signed, written IRB-approved informed consent form
Exclusion Criteria:
- New York Heart Association Class III or IV cardiac disease, or myocardial infarction, severe unstable angina, coronary/peripheral artery bypass graft, congestive heart failure within the past 6 months
- Have a corrected QT interval (using Fridericia's correction formula) (QTcF) of >470 msec (females) and >450 msec (males)
- Active, uncontrolled bacterial, viral, or fungal infections, requiring systemic therapy
- Active, poorly controlled autoimmune or inflammatory diseases
Sites / Locations
- University of Southern CaliforniaRecruiting
- Cedars-Sinai Medical CenterRecruiting
- Northwestern UniversityRecruiting
- Atlantic Health System HospitalRecruiting
Arms of the Study
Arm 1
Arm Type
Experimental
Arm Label
Dose escalation (Q702)
Arm Description
Participants will receive escalating doses of Q702
Outcomes
Primary Outcome Measures
Maximum tolerated dose (MTD), the dose limiting toxicities (DLT) and the safety profile of Q702
Secondary Outcome Measures
Change in the area under curve (AUC) of Q702
Change in the maximum plasma concentration (Cmax) of Q702
Change in the time of maximum plasma concentration (Tmax) of Q702
Tumor response using RECIST version 1.1 throughout study
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT04648254
Brief Title
Oral Axl/Mer/CSF1R Selective Tyrosine Kinase Inhibitor in Patients With Advanced Solid Tumor
Official Title
A Phase 1, Multicenter, Open-label, Dose- Escalation, Safety, Pharmacodynamic, Pharmacokinetic Study of Q702 With a Cohort Expansion at the RP2D in Patients With Advanced Solid Tumors
Study Type
Interventional
2. Study Status
Record Verification Date
September 2022
Overall Recruitment Status
Recruiting
Study Start Date
November 18, 2020 (Actual)
Primary Completion Date
July 18, 2023 (Anticipated)
Study Completion Date
November 18, 2023 (Anticipated)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Sponsor
Name of the Sponsor
Qurient Co., Ltd.
4. Oversight
Studies a U.S. FDA-regulated Drug Product
Yes
Studies a U.S. FDA-regulated Device Product
No
5. Study Description
Brief Summary
This is a Phase 1, open-label, multicenter, dose-escalation, safety, tolerability, pharmacokinetic and pharmacodynamic study with cohort expansion at the RP2D to evaluate safety and anti- tumor activity of Q702 administered orally.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Solid Tumor, Advanced Cancer, Metastatic Cancer
7. Study Design
Primary Purpose
Treatment
Study Phase
Phase 1
Interventional Study Model
Single Group Assignment
Masking
None (Open Label)
Allocation
N/A
Enrollment
78 (Anticipated)
8. Arms, Groups, and Interventions
Arm Title
Dose escalation (Q702)
Arm Type
Experimental
Arm Description
Participants will receive escalating doses of Q702
Intervention Type
Drug
Intervention Name(s)
Q702
Intervention Description
The study drug Q702 will be administered once daily by mouth on Days 1 through 7 and Days 15 through 21 of every treatment cycle.
Primary Outcome Measure Information:
Title
Maximum tolerated dose (MTD), the dose limiting toxicities (DLT) and the safety profile of Q702
Time Frame
28 days of cycle 1
Secondary Outcome Measure Information:
Title
Change in the area under curve (AUC) of Q702
Time Frame
Cycle 1, Days 1,2,8,15,21,22; Cycle 2, Days 1,8,15,22
Title
Change in the maximum plasma concentration (Cmax) of Q702
Time Frame
Cycle 1, Days 1,2,8,15,21,22; Cycle 2, Days 1,8,15,22
Title
Change in the time of maximum plasma concentration (Tmax) of Q702
Time Frame
Cycle 1, Days 1,2,8,15,21,22; Cycle 2, Days 1,8,15,22
Title
Tumor response using RECIST version 1.1 throughout study
Time Frame
Baseline up to approximately 2 years
10. Eligibility
Sex
All
Minimum Age & Unit of Time
18 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
Patients with histologically or cytologically confirmed advanced or metastatic solid tumors, that have progressed following standard of care therapy or for which there is no standard therapy which confers clinical benefit
Measurable disease per RECIST v 1.1
ECOG performance status 0 or 1
Life expectancy of at least 3 months
Age ≥ 18 years
Signed, written IRB-approved informed consent form
Exclusion Criteria:
New York Heart Association Class III or IV cardiac disease, or myocardial infarction, severe unstable angina, coronary/peripheral artery bypass graft, congestive heart failure within the past 6 months
Have a corrected QT interval (using Fridericia's correction formula) (QTcF) of >470 msec (females) and >450 msec (males)
Active, uncontrolled bacterial, viral, or fungal infections, requiring systemic therapy
Active, poorly controlled autoimmune or inflammatory diseases
Central Contact Person:
First Name & Middle Initial & Last Name or Official Title & Degree
Qurient Clinical Trial Information
Phone
+82-31-8060-1610
Ext
(KST)
Email
clinicaltrial_info@qurient.com
Facility Information:
Facility Name
University of Southern California
City
Los Angeles
State/Province
California
ZIP/Postal Code
90033
Country
United States
Individual Site Status
Recruiting
Facility Contact:
First Name & Middle Initial & Last Name & Degree
See Central Contact
Facility Name
Cedars-Sinai Medical Center
City
Los Angeles
State/Province
California
ZIP/Postal Code
90048
Country
United States
Individual Site Status
Recruiting
Facility Contact:
First Name & Middle Initial & Last Name & Degree
See Central Contact
Facility Name
Northwestern University
City
Chicago
State/Province
Illinois
ZIP/Postal Code
60611
Country
United States
Individual Site Status
Recruiting
Facility Contact:
First Name & Middle Initial & Last Name & Degree
See Central Contact
Facility Name
Atlantic Health System Hospital
City
Morristown
State/Province
New Jersey
ZIP/Postal Code
07960
Country
United States
Individual Site Status
Recruiting
Facility Contact:
First Name & Middle Initial & Last Name & Degree
See Central Contact
12. IPD Sharing Statement
Plan to Share IPD
Undecided
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Oral Axl/Mer/CSF1R Selective Tyrosine Kinase Inhibitor in Patients With Advanced Solid Tumor
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