PF-06821497 Treatment Of Relapsed/Refractory SCLC, Castration Resistant Prostate Cancer, and Follicular Lymphoma
Castration Resistant Prostate Cancer (CRPC), Small Cell Lung Cancer (SCLC), Follicular Lymphoma (FL)
About this trial
This is an interventional treatment trial for Castration Resistant Prostate Cancer (CRPC) focused on measuring EZH2, enhancer of zeste homolog 2, castrate resistant prostate cancer, prostatecancer-study.com, CRPC, efficacy, safety, pharmacokinetics, pharmacodynamics, dose escalation, dose expansion, open-label, small cell lung cancer, SCLC, follicular lymphoma, FL, relapsed, refractory
Eligibility Criteria
Key Inclusion Criteria:
Histological or cytological diagnosis of advanced / metastatic solid tumor with the following tumor types in individual study parts:
Part 1A (closed to enrollment):
Part 1B (closed to enrollment):
Part 1C:
• Castration resistant prostate cancer. Patients should have received either abiraterone and/or enzalutamide treatment and have evidence of prostate cancer progression (per PCWG3)
Part 2A:
• Castration resistant prostate cancer. Patients should have received either abiraterone and/or enzalutamide treatment, may have received up to 1 line of chemotherapy and have evidence of prostate cancer progression (per PCWG3)
Part 2B:
- Castration resistant prostate cancer. Patients should have received abiraterone treatment, may have received up to 1 prior line of chemotherapy, have not received prior enzalutamide, and have evidence of prostate cancer progression (per PCWG3)
- Patients must have radiographic evidence of disease
Other inclusion criteria:
- Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) of 0 or 1.
- Adequate organ function
Key Exclusion Criteria:
- Prior Chemotherapy: Part 1C (CRPC): no more than 2 previous regimens of chemotherapy Part 2A: CRPC: no more than 1 previous regimen of systemic chemotherapy Part 2B (CRPC): no more than 1 previous regimen of chemotherapy
- Prior irradiation to >25% of the bone marrow.
- QTcF interval >480 msec at screening.
- Hypertension that cannot be controlled by medications (>150/100 mmHg despite optimal medical therapy).
- Known or suspected hypersensitivity to PF 06821497 or any components or enzalutamide (CRPC)
- Active inflammatory gastrointestinal disease, chronic diarrhea, known diverticular disease or previous gastric resection or lap band surgery. Gastroesophageal reflux disease under treatment with proton pump inhibitors is allowed.
- Current use or anticipated need for food or drugs that are known strong CYP3A4/5 inducers or inhibitors, including their administration within 10 days or 5 half lives of the CYP3A4/5 inhibitor, whichever is longer prior to first dose of investigational product.
Sites / Locations
- Urological Associates of Southern Arizona, P.C .Recruiting
- Banner-University Medical Center Tucson
- The University of Arizona Cancer Center-North Campus
- The University of Arizona Cancer Center
- Urological Associates of Southern Arizona, PCRecruiting
- Pacific Cancer Medical Center INCRecruiting
- City of Hope (City of Hope National Medical Center, City of Hope Medical Center)
- City of Hope Investigational Drug Services (IDS)
- Norwalk HospitalRecruiting
- Illinois CancerCare, P.C.Recruiting
- The University of Kansas Cancer Center, Investigational Drug Services
- The University of Kansas Clinical Research Center
- The University of Kansas Hospital
- The University of Kansas Medical Center Medical Office Building
- The University of Kansas Cancer Center - Indian Creek Campus
- The University of Kansas Cancer Center
- Norton Cancer Institute Pharmacy, Downtown Pharmacy
- Norton Cancer Institute Pharmacy
- Norton Cancer Institute, Norton Healthcare Pavilion
- Norton Hospital
- Maryland Oncology Hematology, P.A.
- Brigham and Women's HospitalRecruiting
- Dana Farber Cancer InstituteRecruiting
- Oncology Hematology West, PC dba Nebraska Cancer SpecialistsRecruiting
- Hackensack University Medical CenterRecruiting
- John Theurer Cancer Center at Hackensack University Medical CenterRecruiting
- OU Medical Center Presbyterian TowerRecruiting
- Stephenson Cancer CenterRecruiting
- Carolina Urologic Research CenterRecruiting
- Parkway Surgery CenterRecruiting
- Tennessee Oncolgy, PLLCRecruiting
- Tennessee Oncology, PLLCRecruiting
- The Sarah Cannon Research InstituteRecruiting
- Texas Oncology - Austin Midtown
- University of Texas Southwestern Medical Center - Simmons Cancer CenterRecruiting
- University of Texas Southwestern Medical Center-Simmons Cancer Center PharmacyRecruiting
- UT Southwestern Medical CenterRecruiting
- UT Southwestern Simmons Cancer CenterRecruiting
- UT Southwestern University Hospital - William P. Clements, JrRecruiting
- UT Southwestern University Hospital - Zale LipshyRecruiting
- Texas Oncology -Fort Worth Cancer Center
- US Oncology Investigational Product Center (IPC)
- US Oncology Investigational Product Center (IPC)
- US Oncology Investigational Products Center
- NEXT Oncology
- Virginia Cancer Specialists, PCRecruiting
- Virginia Oncology Associates
- Seattle Cancer Care AllianceRecruiting
- Specialized Hospital for Active Treatment of Oncology - Haskovo
- Complex Oncology Center - Ruse EOODRecruiting
- "Complex Oncology Center - Vratsa" EOOD
- The First Affiliated Hospital of Guangzhou Medical UniversityRecruiting
- Hunan Cancer HospitalRecruiting
- Zhongda Hospital Southeast UniversityRecruiting
- West China Hospital, Sichuan University
- West China Hospital, Sichuan UniversityRecruiting
- The First Affiliated Hospital of Wenzhou Medical UniversityRecruiting
- National Cancer Center Hospital EastRecruiting
- National Cancer CenterRecruiting
- Seoul National University Bundang HospitalRecruiting
- Seoul National University HospitalRecruiting
- Severance Hospital, Yonsei University Health SystemRecruiting
- Asan Medical CenterRecruiting
- Gangnam Severance Hospital, Yonsei University Health SystemRecruiting
- Samsung Medical CenterRecruiting
- Ewha Womans University Mokdong HospitalRecruiting
- Kyungpook National University Chilgok HospitalRecruiting
- Chungnam national university hospitalRecruiting
- Centrum Medyczne MEDYK
- Centrum Medyczne MEDYKRecruiting
- LUX MED Onkologia Sp. z o.o. Szpital Szamocka
- Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w WarszawieRecruiting
- Private Medical Institution "Euromedservice"
- Private Healthcare Institution "Clinical hospital "RZD-Medicine" of Saint-Petersburg
- Private medical institution "Euromedservice"
- LLC "Neyro-klinika"
- Moscow GBUZ "City clinical hospital n. a. S.P. Botkina" of Moscow health department
- SBHI of Moscow City Clinical Hospital
- Budgetary Healthcare Institution of Omsk region "Clinical Oncological Dispensary"
- Federal State Budgetary Institution National Medical Research Center n.a. V.A. Almazov
- Saint Petersburg State Budgetary Healthcare Institution "City Clinical Oncological Dispensary"
- Non-governmental Healthcare Institution ¨Railway Clinical Hospital of JSC ¨Russian Railways¨
- Private Healthcare Institution "Clinical hospital "RZD-Medicine" of Saint-Petersburg
- Federal State Budgetary Institution National Medical Research Center for Oncology n.a. N.N.
- State Budgetary Healthcare Institution of the Yaroslavl Region
- Institut Català d´Oncología (ICO)-H. Durán i ReynalsRecruiting
- Hospital HM Nou Delfos
- Hospital Universitari Vall d'HebronRecruiting
- Hospital Clinic de BarcelonaRecruiting
- Hospital de la Santa Creu i Sant Pau
- Consorcio Hospitalario Provincial de CastellonRecruiting
- Hospital Universitario Ramon y CajalRecruiting
- H.U. Fundación Jiménez DíazRecruiting
- Hospital Universitario 12 De OctubreRecruiting
- Hospital Universitario HM SanchinarroRecruiting
- Hospital Universitario Virgen de la VictoriaRecruiting
- Hospital Universitari i Politecnic La FeRecruiting
Arms of the Study
Arm 1
Arm 2
Arm 3
Arm 4
Arm 5
Arm 6
Arm 7
Experimental
Experimental
Experimental
Experimental
Experimental
Experimental
Experimental
Dose Escalation (Part 1A)
Dose Escalation (Part 1B)
Dose Escalation (Part 1C)
Dose Escalation (Part 2A)
Dose Expansion (Part 2B)
Japan Cohort
China cohort
Participants with SCLC, CRPC and FL will receive PF-06821497 at escalating dose levels
Participants with FL will receive PF-06821497 at escalating dose levels
Participants with CRPC will receive PF-06821497 at escalating dose levels.
Participants with CRPC and SCLC will receive PF-06821497 at escalating dose levels in combination with SOC.
Participants with CRPC will receive PF-06821497 in combination with SOC or SOC alone.
Participants with CRPC will receive PF-06821497 at one or two doses
Participants will receive PF-06821497 at one or two doses