Probenecid as Medication for Alcohol Use Disorder (PROB)
Primary Purpose
Alcohol Use Disorder
Status
Recruiting
Phase
Phase 1
Locations
United States
Study Type
Interventional
Intervention
Probenecid
Matching placebo
Sponsored by
About this trial
This is an interventional other trial for Alcohol Use Disorder
Eligibility Criteria
Inclusion Criteria:
- Male or female, 21-70 (inclusive) years; women >7 drinks/week; men >14 drinks/week;
- meet any DSM-5 criteria score for AUD;
- Breath alcohol Content (BrAC)=0.00 at each visit;
- In good health as confirmed by medical history, physical examination and lab tests;
- Willing to adhere to the study procedures;
- Understand informed consent and questionnaires in English at an 8th grade level
Exclusion Criteria:
- Women who are breastfeeding or have a positive urine screen for pregnancy
- CrCl < 60mL/min
- Taking aspirin (salicylates may reduce effect of probenecid)
- Taking penicillin
- Taking methotrexate (may increase concentration)
- Taking other medications that may interact with probenecid
- History of suicide attempts in the last three years
- Current diagnosis of another substance disorder(s) other than nicotine, as assessed by self-reports and urine toxicology screen at baseline
- History of hypersensitivity to sulfa drugs
Sites / Locations
- Brown UniversityRecruiting
Arms of the Study
Arm 1
Arm 2
Arm Type
Experimental
Placebo Comparator
Arm Label
Probenecid
matching placebo
Arm Description
2g probenecid, one pill by mouth once, for one day
Placebo, one pill by mouth once, for one day
Outcomes
Primary Outcome Measures
Stimulant effects of alcohol when co-administered with drug or matching placebo
assessed using the change in the Biphasic Alcohol Effects Scale (BAES), scale 0-10 (direct and reverse score)
Secondary Outcome Measures
Sedative effects of alcohol when co-administered with drug or matching placebo
assessed using change in the Biphasic Alcohol Effects Scale (BAES), scale 0-10 (direct and reverse score)
Alcohol craving
assessed using change in the alcohol urge questionnaire (AUQ), scale 0-7 (7 worse outcome)
Full Information
1. Study Identification
Unique Protocol Identification Number
NCT04218357
Brief Title
Probenecid as Medication for Alcohol Use Disorder
Acronym
PROB
Official Title
Probenecid as Pharmacotherapy for Alcohol Use Disorder
Study Type
Interventional
2. Study Status
Record Verification Date
July 2023
Overall Recruitment Status
Recruiting
Study Start Date
December 2, 2020 (Actual)
Primary Completion Date
December 20, 2023 (Anticipated)
Study Completion Date
December 20, 2023 (Anticipated)
3. Sponsor/Collaborators
Responsible Party, by Official Title
Principal Investigator
Name of the Sponsor
Brown University
4. Oversight
Studies a U.S. FDA-regulated Drug Product
Yes
Studies a U.S. FDA-regulated Device Product
No
Product Manufactured in and Exported from the U.S.
Yes
Data Monitoring Committee
No
5. Study Description
Brief Summary
The design is a randomized, within-subject, crossover, double-blind, placebo-controlled human alcohol laboratory study with one oral dose of 2g probenecid or placebo administered in two laboratory sessions.
Detailed Description
There will be a total of four study visits. Visit 1 is the screening for eligibility (medical and physical examination). On Visits 2 and 3, participants will undergo an alcohol laboratory session with a one week washout period before administering the alternate therapy. The study will conclude at Visit 4.
6. Conditions and Keywords
Primary Disease or Condition Being Studied in the Trial, or the Focus of the Study
Alcohol Use Disorder
7. Study Design
Primary Purpose
Other
Study Phase
Phase 1
Interventional Study Model
Crossover Assignment
Masking
ParticipantCare ProviderInvestigatorOutcomes Assessor
Allocation
Randomized
Enrollment
34 (Anticipated)
8. Arms, Groups, and Interventions
Arm Title
Probenecid
Arm Type
Experimental
Arm Description
2g probenecid, one pill by mouth once, for one day
Arm Title
matching placebo
Arm Type
Placebo Comparator
Arm Description
Placebo, one pill by mouth once, for one day
Intervention Type
Drug
Intervention Name(s)
Probenecid
Other Intervention Name(s)
Probalan
Intervention Description
safety
Intervention Type
Drug
Intervention Name(s)
Matching placebo
Other Intervention Name(s)
Placebo
Intervention Description
Placebo
Primary Outcome Measure Information:
Title
Stimulant effects of alcohol when co-administered with drug or matching placebo
Description
assessed using the change in the Biphasic Alcohol Effects Scale (BAES), scale 0-10 (direct and reverse score)
Time Frame
Change from Day 3 to day 10 of the trial
Secondary Outcome Measure Information:
Title
Sedative effects of alcohol when co-administered with drug or matching placebo
Description
assessed using change in the Biphasic Alcohol Effects Scale (BAES), scale 0-10 (direct and reverse score)
Time Frame
Change from Day 3 to day 10 of the trial
Title
Alcohol craving
Description
assessed using change in the alcohol urge questionnaire (AUQ), scale 0-7 (7 worse outcome)
Time Frame
Change from Day 3 to day 10 of the trial
10. Eligibility
Sex
All
Minimum Age & Unit of Time
21 Years
Maximum Age & Unit of Time
70 Years
Accepts Healthy Volunteers
No
Eligibility Criteria
Inclusion Criteria:
Male or female, 21-70 (inclusive) years; women >7 drinks/week; men >14 drinks/week;
meet any DSM-5 criteria score for AUD;
Breath alcohol Content (BrAC)=0.00 at each visit;
In good health as confirmed by medical history, physical examination and lab tests;
Willing to adhere to the study procedures;
Understand informed consent and questionnaires in English at an 8th grade level
Exclusion Criteria:
Women who are breastfeeding or have a positive urine screen for pregnancy
CrCl < 60mL/min
Taking aspirin (salicylates may reduce effect of probenecid)
Taking penicillin
Taking methotrexate (may increase concentration)
Taking other medications that may interact with probenecid
History of suicide attempts in the last three years
Current diagnosis of another substance disorder(s) other than nicotine, as assessed by self-reports and urine toxicology screen at baseline
History of hypersensitivity to sulfa drugs
Central Contact Person:
First Name & Middle Initial & Last Name or Official Title & Degree
Zoe Brown, BA
Phone
401-863-6646
Email
alcohol-stress-study@brown.edu
Overall Study Officials:
First Name & Middle Initial & Last Name & Degree
Carolina L Haass-Koffler, PHARMD
Organizational Affiliation
Brown University
Official's Role
Principal Investigator
Facility Information:
Facility Name
Brown University
City
Providence
State/Province
Rhode Island
ZIP/Postal Code
20923
Country
United States
Individual Site Status
Recruiting
Facility Contact:
First Name & Middle Initial & Last Name & Degree
Zoe Brown
Phone
401-863-6646
First Name & Middle Initial & Last Name & Degree
Carolina Haass-Koffler, PHARMD
12. IPD Sharing Statement
Plan to Share IPD
No
Citations:
PubMed Identifier
31535696
Citation
Tunstall BJ, Lorrai I, McConnell SA, Gazo KL, Zallar LJ, de Guglielmo G, Hoang I, Haass-Koffler CL, Repunte-Canonigo V, Koob GF, Vendruscolo LF, Sanna PP. Probenecid Reduces Alcohol Drinking in Rodents. Is Pannexin1 a Novel Therapeutic Target for Alcohol Use Disorder? Alcohol Alcohol. 2019 Jan 9;54(5):497-502. doi: 10.1093/alcalc/agz054.
Results Reference
result
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Probenecid as Medication for Alcohol Use Disorder
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